阿戈美拉汀
- 价格: ¥99/瓶
- 发布日期: 2019-04-01
- 更新日期: 2025-10-15
产品详请
| 产地 |
加拿大
|
| 品牌 |
进口
|
| 货号 |
01-430000
|
| 包装规格 |
10mg,100mg
|
| 纯度 |
98%
|
| CAS编号 |
138112-76-2
|
| 别名 |
N-[2-(7-Methoxy-1-naphthalenyl)ethyl]acetamide; N-[2-(7-Methoxy-1-naphthyl)
ethyl]acetamide; S 20098; Valdoxan;
|
货号:01-430000
中文名称:阿戈美拉汀
英文名称:Agomelatine-d4
CAS号:138112-76-2
重量:10mg
重量:100mg
分子式:C15H17NO2
别名:N-[2-(7-Methoxy-1-naphthalenyl)ethyl]acetamide; N-[2-(7-Methoxy-1-naphthyl)
ethyl]acetamide; S 20098; Valdoxan;
应用介绍:Agomelatine is a melatoninergic agonist and selective antagonist of 5-HT2C receptors, and has been shown to be active in several animal models of depression. Agomelatine (S20098) displayed pKi values of 6.4 and 6.2 at native (porcine) and cloned, human (h)5-hydroxytryptamine (5-HT)2C receptors, respectively.